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Development of CRF₁ receptor antagonists as antidepressants and anxiolytics: Progress to dateVALDEZ, Glenn R.CNS drugs. 2006, Vol 20, Num 11, pp 887-896, issn 1172-7047, 10 p.Article

Stress and central Urocortin increase anxiety-like behavior in the social interaction test via the CRF₁ receptorGEHLERT, Donald R; SHEKHAR, Anantha; MORIN, S. Michelle et al.European journal of pharmacology. 2005, Vol 509, Num 2-3, pp 145-153, issn 0014-2999, 9 p.Article

An arginine vasopressin V_1b antagonist, SSR149415 elicits antidepressant-like effects in an olfactory bulbectomy modelIIJIMA, Michihiko; CHAKI, Shigeyuki.Progress in neuro-psychopharmacology & biological psychiatry. 2007, Vol 31, Num 3, pp 622-627, issn 0278-5846, 6 p.Article

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NBI 30775 (R121919), an orally active antagonist of the corticotropin-releasing factor (CRF) type-1 receptor for the treatment of anxiety and depressionCHEN CHEN; GRIGORIADIS, Dimitri E.Drug development research. 2005, Vol 65, Num 4, pp 216-226, issn 0272-4391, 11 p.Article

Binding differences of human and amphibian corticotropin-releasing factor type 1 (CRF1) receptors: identification of amino acids mediating high-affinity astressin binding and functional antagonismDAUTZENBERG, Frank M; WILLE, Sandra.Regulatory peptides. 2004, Vol 118, Num 3, pp 165-173, issn 0167-0115, 9 p.Article

Control by tachykinin NK₂ receptors of CRF₁ receptor-mediated activation of hippocampal acetylcholine release in the rat and guinea-pigDESVIGNES, C; ROUQUIER, L; SOUILHAC, J et al.Neuropeptides (Edinburgh). 2003, Vol 37, Num 2, pp 89-97, issn 0143-4179, 9 p.Article

Urocortin promotes the development of vasculitis in a rat model of thromboangiitis obliterans via corticotrophin-releasing factor type 1 receptorsYOUHUA XU; RONGJIAN ZHANG; YUANYUAN GUO et al.British journal of pharmacology. 2009, Vol 157, Num 8, pp 1368-1379, issn 0007-1188, 12 p.Article

The role of CRF₁ receptors for sympathetic nervous response to laparotomy in anesthetized ratsUETSUKI, Nobuo; SEGAWA, Hajime; MAYAHARA, Taku et al.Brain research. 2005, Vol 1044, Num 1, pp 107-115, issn 0006-8993, 9 p.Article

Blockade of the Corticotropin Releasing Factor Type 1 Receptor Attenuates Elevated Ethanol Drinking Associated With Drinking in the Dark ProceduresSPARTA, Dennis R; SPARROW, Angela M; LOWERY, Emily G et al.Alcoholism, clinical and experimental research. 2008, Vol 32, Num 2, pp 259-265, issn 0145-6008, 7 p.Article

CORTICOTROPIN RELEASING FACTOR-1 RECEPTOR ANTAGONIST, CP-154,526, BLOCKS THE EXPRESSION OF ETHANOL-INDUCED BEHAVIORAL SENSITIZATION IN DBA/2J MICEFEE, J. R; SPARTA, D. R; PICKER, M. J et al.Neuroscience. 2007, Vol 150, Num 1, pp 14-21, issn 0306-4522, 8 p.Article

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Differential profile of CRF receptor distribution in the rat stomach and duodenum assessed by newly developed CRF receptor antibodiesCHATZAKI, Ekaterini; MURPHY, Brian J; LIXIN WANG et al.Journal of neurochemistry. 2004, Vol 88, Num 1, pp 1-11, issn 0022-3042, 11 p.Article

MPZP : A novel small molecule corticotropin-releasing factor type 1 receptor (CRF₁) antagonistRICHARDSON, Heather N; ZHAO, Yu; FEKETE, Eva M et al.Pharmacology, biochemistry and behavior. 2008, Vol 88, Num 4, pp 497-510, issn 0091-3057, 14 p.Article

Dependence-induced increases in ethanol self-administration in mice are blocked by the CRF₁ receptor antagonist antalarmin and by CRF₁ receptor knockoutCHU, Kathleen; KOOB, George F; COLE, Maury et al.Pharmacology, biochemistry and behavior. 2007, Vol 86, Num 4, pp 813-821, issn 0091-3057, 9 p.Article

A 6-Week Randomized, Placebo-Controlled Trial of CP-316,311 (a Selective CRH₁ Antagonist) in the Treatment of Major DepressionBINNEMAN, Brendon; FELTNER, Douglas; KOLLURI, Sheela et al.The American journal of psychiatry. 2008, Vol 165, Num 5, pp 617-620, issn 0002-953X, 4 p.Article

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